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Tlhahiso ea Lihlahisoa 99% Purity White Powder Antitumor Polypeptide Pharma Mophato oa Lipatlisiso tsa Kankere MELITTIN CAS 20449-79-0

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Melittin, peptide e amanang le 'mele ea ho itšireletsa mafung ea PLA2 e tsoang mahlokong a linotsi, e eketsa ts'ebetso ea li-enzyme tse boima ba limolek'hule [1].Melittin ke peptide ea cytotoxic e tsoang ho chefo ea linotsi.Melittin e bonts'itse chefo ho lisele tsa A2780CR le A2780 ka bobeli, tse nang le boleng ba IC50 ba 4.5 le 6.8 μg/mL, ka ho latellana.Melittin e na le thepa ea tlhaho ea antibacterial, antiviral le anti-inflammatory.E boetse e bonts'itsoe hore e na le litlamorao tse ngata tsa anticancer meleng e mengata e fapaneng ea mofets'e, ho kenyelletsa le gastric, matsoele, mahe a bomme, sebete, prostate, molomo oa popelo le lisele tsa mofetše oa matšoafo.Melittin, e leng amphipathic hemolytic peptide, e fana ka litlamorao tse ka bang teng tsa anticancer ka ho thibela ho ata ha lisele, ho kenella ha apoptosis le necrosis e tobileng.


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MELITTIN CAS 20449-79-0

Tšebeliso ea MELITTIN CAS 20449-79-0:

Melitin ke motsoako o ka sehloohong o sebetsang oa chefo ea linotsi.Beevenom ke mofuta oa chefo e bonaletsang e nang le monko o monate o hlahisoang ke litšoelesa tsa mahloko a linotši le litšoelesa tse ling.Ha e tlōtsoe, e ntšoa ho hlabang.Har'a likarolo tse ngata tsa mahloko a linotsi, melittin e na le lintho tse phahameng ka ho fetisisa, tse etsang karolo ea 50% ea boima bo omeletseng ba linotši, 'me e na le ts'ebetso e phahameng ea likokoana-hloko.Melittin ke linear peptide e entsoeng ka 26 amino acid, e nang le boima ba molek'hule ea 2849. Melittin e na le ts'ebetso e phahameng ea likokoana-hloko.Lithuto tsa morao-rao tsa meriana li bontšitse hore li na le li-anti-inflammatory, analgesic, inhibiting platelet aggregation, anti-AIDS le liphello tse ling tse ngata.Melittin e ka hlahisa phello e matla ea ho bolaea liseleng tse fapaneng tsa hlahala ka mekhoa e fapaneng, 'me ke setlhare se ts'episang haholo se khahlanong le hlahala.

Melittin e ka thibela kholo le ho ikatisa ha mefuta e fetang 20 ea libaktheria tse ntle tsa gram-positive le tse mpe, hape e ka ntlafatsa katleho ea antibacterial ea sulfonamides le penicillin.Melittin e senya lera la sele ea baktheria ka ho tlama lera ho fihlela sepheo sa bacteriolysis.Ka bobeli melittin le tse tsoang ho eona tse tšeletseng li ka fetola tšebetso ea T lymphocyte tse tšoaelitsoeng ke HIV, tsa thibela ho ikatisa ha HIV, le ho fokotsa tšoaetso ea kokoana-hloko.

  1. Liphello tsa ho bolaea ka kotloloho Liteko tsa in vitro li netefalitse hore melittin e na le phello e hlakileng ea ho bolaea melaleng e fapaneng ea lisele tsa tumor joalo ka osteosarcoma, mofetše oa mahe a bomme le glioma, mme phello ea polao e amana hantle le lethal dose.Melittin e ka bolaea lisele tsa hlahala le ho thibela kholo ea lisele tsa hlahala, 'me ha e na phello e hlakileng ho holeng ha lisele tse tloaelehileng.Melittin e ka kenya ka har'a lisele tsa lisele tsa K562, ea etsa li-pores, e khothalletsa ho phalla ha Ca2 +, ho eketsa khatello ea Ca2 + liseleng, ho baka lisele tsa lysis, le ho bolaea lisele tsa K562 ka ho toba.Ka kakaretso ho lumeloa hore melittin e qhala lera la mitochondrial ea lisele, e thibela tšebetso e tloaelehileng ea phefumoloho ea lisele tsa tumor, e senya matla a bona a ho phefumoloha a aerobic, e thibela kholo ea lisele tsa hlahala, 'me e bolaea lisele tsa hlahala ka kotloloho.
  2. Immunomodulatory effect Ho itšireletsa ha lisele ke ntho ea bohlokoa ea tšireletso bakeng sa 'mele khahlanong le lihlahala le tšoaetso ea kokoana-hloko.Boemo ba ts'ebetso ea 'mele ea' mele ea ho itšireletsa mafung e phetha karolo ea bohlokoa ketsahalong le nts'etsopele ea lihlahala.Ho ntlafatsa ts'ebetso ea 'mele ea ho itšireletsa mafung ho ka bapala phello e itseng ea anti-tumor.
  3. Induction of tumor cell apoptosis Apoptosis, eo hape e tsejoang e le programmed cell death, ke ts'ebetso e sebetsang ea bioloji e laoloang ke mefuta e fapaneng ea liphatsa tsa lefutso.Ka hona, apoptosis ke ts'ebetso e sebetsang, e kenyelletsang ts'ebetso, polelo le taolo ea letoto la liphatsa tsa lefutso.Lithuto tsa sejoale-joale li bonts'itse hore lithethefatsi tse ngata tsa chemotherapeutic li ka fihlela sepheo sa kalafo ka ho kenya apoptosis liseleng tsa mofetše.Hore na ho susumetsa apoptosis e se e le e 'ngoe ea mekhoa ea ho hlahloba lithethefatsi tse thibelang mofetše.

Melittin e ka thibela ts'ebetso ea sPLA2 ho tsoa mehloling e fapaneng, mme sekhahla sa ho thibela ts'ebetso ea sPLA2 ho synovial fluid ea bakuli ba RA se ka fihla ho 96%.Ka hona, tšebeliso ea melittin e ka fokotsa tsoelo-pele ea RA.

Sub-dose melittin e ka fokotsa haholo sekhahla sa lysis sa tlatsetso ho lisele.Mokhoa ona oa tšireletso o ka 'na oa amana le melittin e khothalletsang phallo ea Ca2 +, e susumetsang tsamaiso ea ho fetisetsa lipontšo tsa intracellular le protheine e sireletsang synthesis.Ho khothaletsoa hore tšebeliso ea tekanyo e nepahetseng ea melittin e na le boleng bo itseng ba bongaka kalafong ea RA ke Chemicalbook.Lilemong tsa morao tjena, liphuputso li bontšitse hore likhakanyo tse fapaneng tsa melittin li ka ama ts'ebetso ea lisele ka liteishene tse fapaneng mme tsa ba le litlamorao tse fapaneng tsa tlhaho.Tšebeliso e nepahetseng ea melittin e tla fana ka phekolo e ncha bakeng sa mafu a mang.

MELITTIN CAS 20449-79-0

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