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Ƙirƙirar Ƙirƙirar 99% Tsarkake Farin Foda Antitumor Polypeptide Pharma Grade Cancer Research MELITTIN CAS 20449-79-0

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Category: Abubuwa masu guba

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Melittin, peptide mai haɓaka PLA2 mai alaƙa da rigakafi daga dafin kudan zuma, yana haɓaka ayyukan enzymes masu nauyi masu nauyi [1].Melittin shine peptide cytotoxic wanda aka samo daga dafin kudan zuma.Melittin ya nuna guba ga duka kwayoyin A2780CR da A2780, tare da ƙimar IC50 na 4.5 da 6.8 μg/mL, bi da bi.Melittin yana da na halitta antibacterial, antiviral da anti-mai kumburi Properties.Hakanan an nuna cewa yana da tasirin anticancer da yawa a cikin layukan ƙwayoyin cutar kansa daban-daban, gami da ciki, nono, ovarian, hanta, prostate, mahaifa, da layukan kansar huhu.Melittin, peptide hemolytic amphipathic, yana haifar da tasirin maganin cutar kansa ta hanyar hana yaduwar kwayar halitta, shigar da apoptosis, da necrosis kai tsaye.


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MELITTIN CAS 20449-79-0

MELITTIN CAS 20449-79-0 Amfani:

Melitin shine babban sinadarin dafin kudan zuma.Beevenom wani nau'i ne na dafin dafin da ke da ƙamshi mai ƙamshi wanda ma'aikaci ya ɓoye dafin kudan zuma da gland.Idan aka keta shi, ana fitar da shi daga simintin.Daga cikin nau'ikan dafin kudan zuma da yawa, melittin yana da mafi girman abun ciki, wanda ya kai kusan kashi 50% na busasshen nauyin dafin kudan zuma, kuma yana da babban aikin nazarin halittu.Melittin peptide na layi ne wanda ya ƙunshi amino acid 26, tare da nauyin kwayoyin dangi na 2849. Melittin yana da babban aikin nazarin halittu.Nazarin harhada magunguna na zamani sun nuna cewa yana da maganin kumburi, analgesic, hana haɓakar platelet, anti-AIDS da sauran sakamako masu yawa.Melittin na iya haifar da sakamako mai ƙarfi na kisa akan nau'ikan ƙwayoyin cuta iri-iri ta hanyoyi daban-daban, kuma yana da matukar alƙawarin maganin ƙwayar cuta.

Melittin na iya hana girma da haifuwa fiye da nau'ikan gram 20 na ƙwayoyin cuta masu kyau da marasa kyau, kuma yana iya haɓaka tasirin ƙwayoyin cuta na sulfonamides da penicillins.Melittin yana lalata ƙwayar ƙwayar ƙwayar cuta ta hanyar ɗaure ga membrane don cimma manufar bacteriolysis.Dukansu melittin da abubuwan da suka samo asali guda shida na iya canza aikin T lymphocytes masu kamuwa da kwayar cutar HIV, hana kwafin kwayar cutar HIV, da rage kamuwa da cutar.

  1. Tasirin kisa kai tsaye Gwaje-gwajen vitro sun tabbatar da cewa melittin yana da tasirin kisa na zahiri akan layukan ƙwayoyin cuta daban-daban kamar osteosarcoma, ciwon daji na ovarian, da glioma, kuma tasirin kisan yana da alaƙa da alaƙa da kashi.Melittin na iya kashe ƙwayoyin ƙwayar cuta kuma ya hana haɓakar ƙwayoyin tumor, kuma ba shi da wani tasiri a zahiri ga ci gaban ƙwayoyin al'ada.Melittin na iya sakawa a cikin kwayar halitta ta kwayoyin K562, samar da pores, inganta haɓakar Ca2 +, ƙara yawan taro na Ca2 + a cikin sel, haifar da lysis cell, kuma kai tsaye kashe K562 Kwayoyin.An yi imani da cewa melittin yana narkar da membrane na mitochondrial na sel, yana hana aikin numfashi na al'ada na ƙwayoyin tumor, yana lalata ƙarfin numfashin su, yana hana ci gaban ƙwayar ƙwayar cuta, kuma yana kashe ƙwayoyin tumor kai tsaye.
  2. Immunomodulatory Tasirin rigakafi na kwayar halitta muhimmin abu ne na kariya ga jiki daga ciwace-ciwacen daji da cututtukan hoto.Halin aikin rigakafi na salula yana taka muhimmiyar rawa wajen faruwa da ci gaban ciwace-ciwacen daji.Haɓaka aikin rigakafi na salula na iya taka wani tasirin anti-tumor.
  3. Ƙaddamar da ƙwayar ƙwayar cuta apoptosis Apoptosis, wanda kuma aka sani da tsarin mutuwa tantanin halitta, wani tsari ne na kwayoyin halitta mai aiki wanda ke sarrafa nau'ikan kwayoyin halitta.Sabili da haka, apoptosis wani tsari ne mai aiki, wanda ya haɗa da kunnawa, magana da tsari na jerin kwayoyin halitta.Nazarin zamani ya nuna cewa yawancin magungunan chemotherapeutic na iya cimma manufar warkewa ta hanyar haifar da apoptosis a cikin kwayoyin cutar kansa.Ko haifar da apoptosis ya zama ɗaya daga cikin ma'auni don tantance magungunan anticancer.

Melittin na iya hana ayyukan sPLA2 daga maɓuɓɓuka daban-daban, kuma ƙimar hana sPLA2 a cikin ruwan synovial na marasa lafiya na RA na iya kaiwa 96%.Saboda haka, aikace-aikacen melittin na iya rage ci gaban RA.

Sub-dose melittin na iya rage yawan lysis na haɓaka ga sel.Wannan tsarin kariya yana iya kasancewa yana da alaƙa da melittin yana haɓaka kwararar Ca2+, yana ƙarfafa tsarin watsa siginar ciki da haɗin haɗin furotin mai karewa.An ba da shawarar cewa aikace-aikacen adadin melittin da ya dace yana da takamaiman ƙimar asibiti a cikin maganin RA ta Chemicalbook.A cikin 'yan shekarun nan, binciken ya nuna cewa nau'i-nau'i daban-daban na melittin na iya rinjayar ayyukan tantanin halitta ta hanyoyi daban-daban da kuma haifar da nau'o'in ilimin halitta.Yin amfani da melittin da ya dace zai samar da sababbin jiyya ga wasu cututtuka.

MELITTIN CAS 20449-79-0

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