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GHRP-6 CAS: 87616-84-0 Kukura kwehomoni kuburitsa peptide

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  • CAS NO:87616-84-0
  • Zita:GHRP-6
  • Melting point:>160o C (Zvita.)
  • Boiling point:1407.0±65.0 °C(Zvakafanotaurwa)
  • Chemical formula:C 46 H 56 N 12 O 6
  • density1.333±0.06 g/cm3(Zvakafanotaurwa)
  • kuchengetedza temp.:−20°C
  • pka:13.42±0.46(Zvakafanotaurwa)
  • fomu:Solid
  • Molar mass:873.032
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  • Product Detail

    Product Tags

    Usage

    Growth hormone-releasing peptide 6 (GHRP-6) (developmental code name SKF-110679), inozivikanwawo sekukura hormone-releasing hexapeptide, ndeimwe yezvakati wandei synthetic met-enkephalin analogues anosanganisira asiri echisikigo D-amino acids, akagadzirirwa avo. kukura kwehomoni-kuburitsa basa uye inonzi kukura kwehomoni secretagogues.Ivo havana basa reopioid asi vane simba vanosimudzira kukura kwehomoni kuburitswa.Aya ma secretagogue akasiyana nekukura kwehomoni kuburitsa mahormone mukuti ivo havagovane hukama hwekutevedzana uye vanowana basa ravo kuburikidza ne activation yeyakasiyana receptor.Iyi receptor pakutanga yainzi kukura kwehomoni secretagogue receptor, asi nekuda kwekuzowanikwa kwakazotevera, iyo hormone ghrelin yave kunzi receptor's natural endogenous ligand, uye yakatumidzwa zita rekuti ghrelin receptor.Naizvozvo, aya maGHSR agonist anoita seanogadzira ghrelin mimetics.

    Zvakaonekwa kuti kana GHRP-6 uye insulin inoshandiswa panguva imwe chete, mhinduro yeGH kuGHRP-6 inowedzera.Nekudaro, kudyiwa kwemacarbohydrates uye / kana mafuta ekudya, kutenderedza hwindo rekutonga reGH secretagogues zvakanyanya blunts kuburitswa kweGH.Ongororo yechangobva kuitika mumakonzo akajairwa yakaratidza misiyano yakakura mukuumbwa kwemuviri, kukura kwemisumbu, glucose metabolism, chiyeuchidzo uye basa remoyo mumakonzo ari kupihwa GHRP-6.Pachine mibvunzo mizhinji maererano nekomboni iyi itsva.

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