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Anti-Estrogen Yogwira Ntchito Exemestane / Aromasin Powder Kuti Mupeze Minofu CAS 107868-30-4

Kufotokozera mwachidule:

Kufotokozera Mwatsatanetsatane Zamalonda

Dzina Lina:Aromasin
MF:C20H24O2
MW:296.4
MP:155.13°C
Nthawi Yosungira:Sungani Pa -20 ° C
Ntchito:Anti-Estrogen
Maonekedwe:Ufa Wakristalo Woyera, Wopanda fungo
Kuwala Kwakukulu:Anti Estrogen Products, Anti Estrogen Mankhwala


Tsatanetsatane wa Zamalonda

Zolemba Zamalonda

Exemestane (Aromasin)Zambiri Zamalonda

Dzina lazogulitsa: Exemestane
Mawu ofanana: Aromasin
CAS: 107868-30-4
MF: C20H24O2
MW: 296.4
mp: 155.13°C
kutentha kosungira: Sungani pa -20°C
maonekedwe: ufa wonyezimira woyera mpaka wachikasu

Kufotokozera:
Aromasin amagwiritsidwa ntchito kulimbana ndi khansa ya m'mawere ndikukweza testosterone m'thupi.
Exemestane imalepheretsa njira ya aromatisation.Choncho amachepetsa kuchuluka kwa estrogen m'thupi.Kumayambiriro kwa khansa ya m'mawere, kutenga exemestane kungathandize kuletsa khansa ya m'mawere kubwerera.Mu khansa ya m'mawere yapita patsogolo maselo a khansa amatha kukula pang'onopang'ono kapena kusiya kukula kwathunthu.
Exemestane ndi aromatase inhibitor.Izi zikutanthauza kuti imalepheretsa enzyme aromatase (yomwe imapezeka mu minofu ya thupi, khungu, chifuwa ndi mafuta), yomwe imagwiritsidwa ntchito potembenuza androgens (mahomoni opangidwa ndi adrenal glands) kukhala estrogen.Ngati estrogen palibe, zotupa zomwe zimadalira hormone iyi kuti zikule zimachepa

Chitsanzo (1)

Kugwiritsa ntchito Exemestane (Aromasin).

Amagwiritsidwa ntchito pochiza khansa ya m'mawere ya metastatic ndipo amagwiritsidwa ntchito ngati chithandizo pochiza khansa ya m'mawere oyambirira.

1. Ndi imodzi mwa mankhwala amphamvu kwambiri opondereza estrogen.
2. Ndi imodzi mwazinthu zabwino kwambiri zochepetsera kununkhira kwa ma steroid.
3. Imapezeka kwa omanga thupi omwe amatenga anabolic steroids.
4. Imachita mwa kutsekereza enzyme aromatase, kenako ndikuletsa kupanga kwa estrogen.
5. Ndi mtundu wa antineoplastic (hormonal) zopangira.

Exemestane (Aromasin)Mapulogalamu

Aromasin amagwiritsidwa ntchito kulimbana ndi khansa ya m'mawere ndikukweza testosterone m'thupi.
Exemestane acetate imatchinga njira ya aromatisation.Choncho amachepetsa kuchuluka kwa estrogen m'thupi.Kumayambiriro kwa khansa ya m'mawere, kutenga exemestane acetate kungathandize kuletsa khansa ya m'mawere kubwerera.Mu khansa ya m'mawere yapita patsogolo maselo a khansa amatha kukula pang'onopang'ono kapena kusiya kukula kwathunthu.

Ambiri aromatase inhibitors si steroids mu mawonekedwe aliwonse kapena mawonekedwe koma apa tiyenera kupanga zosiyana.Mvetsetsani, ambiri omwe amagula Aromasin amatero chifukwa kugwiritsa ntchito kwake ndi ma steroids ena nthawi zambiri kumakhala kofunika kwambiri pokhudzana ndi zotsatirapo zake koma Aromasin yokha imakhala ndi mikhalidwe ina ya androgenic.Ngakhale zili choncho, pokhala ndi chikhalidwe cha androgenic ndi kuchepetsa estrogen yomwe timakhudzidwa nayo kwambiri.

m'badwo wachitatu aromatase inhibitors, omwe amagwiritsidwa ntchito pochiza khansa ya m'mawere ya metastatic ndipo amagwiritsidwa ntchito ngati chithandizo pochiza khansa ya m'mawere yoyambirira.
Makhansa ambiri am'mawere amalimbikitsidwa kukula ndi mahomoni ogonana achikazi estrogen ndi progesterone.Makhansa a m'mawerewa amatchedwa "hormone sensitive" kapena "hormone receptor positive" ndipo amatha kuchiritsidwa ndi mankhwala omwe amaletsa zotsatira za mahomoniwa.

Kwa amayi omwe asiya kusamba, estrogen imapangidwa makamaka mwa kusintha ma androgens (mahomoni ogonana opangidwa ndi adrenal glands) kukhala oestrogens.Njirayi imatchedwa aromatisation ndipo imachitika makamaka mumafuta, minofu ndi khungu.Zimafunika puloteni inayake yotchedwa aromatase.
Aromasin imalepheretsa kununkhira.Choncho amachepetsa kuchuluka kwa estrogen m'thupi.Kumayambiriro kwa khansa ya m'mawere, kutenga Aromasin kungathandize kuti khansa ya m'mawere ibwererenso.Mu khansa ya m'mawere yapita patsogolo maselo a khansa amatha kukula pang'onopang'ono kapena kusiya kukula kwathunthu.

Chitsanzo (4)
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