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Imodyuli ye-Androgen receptor S-4(Andarine)

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I-S-4 (i-Andarine) i-modulator ye-androgen receptor ekhethiweyo.Igama layo elipheleleyo ngu-S-40503, okanye i-S-4 ngokufutshane, kwaye igama layo lokurhweba yi-Andarine, eyaphuhliswa yinkampani yaseJapan yamayeza i-KakenPharmaceuticals njengonyango lwe-osteoporosis.I-S-4 isebenza ngokufanayo kwi-steroids Conlillon kunye ne-Oxyandrosaurus, kodwa ayisiyiyo i-steroid.

 

Umsebenzi kunye neempawu ze-S-4 (Andarine)

Umsebenzi kunye neempawu ze-S-4 (i-Andarine) i-S-4 inobudlelwane obuqinileyo kunye ne-androgen receptors yethambo kunye ne-muscle, kwaye idigri yokubopha ihle kakhulu.Nangona ingabangeli isihlunu esikhulu kunye nokuzuza ubunzima okwenziwa yiQunbolone, inefuthe elimangalisayo ekulahlekeni kwamafutha.Ngoba?I-S-4 ine-index ephezulu ye-androgen kunye ne-anabolism ephantsi kakhulu yeemveliso ze-SARMS, kwaye xa i-androgens inamathele kwi-androgen receptors kwi-adipose tissue okanye i-fat (esinayo kunye ne-fat) ibangela i-oxidation ye-fat.

Le SARM ikhethiweyo kwaye ayinayo umsebenzi obalulekileyo we-prostatic.I-S-4 inefuthe elibi ekukhuleni kwezihlunu kwiidosi ezisezantsi kwaye ngokuqhelekileyo idinga iidosi ezinkulu ukuze ikhuthaze inzuzo yobunzima bomzimba obuncinci.Njengoko benditshilo ngaphambili, imisebenzi ye-S-4 efana ne-Corylone kunye ne-Oxyandrosaurus, kodwa i-S-4 ayinayo imiphumo echaphazelekayo ye-androgen.

I-SARM iyasebenza ngokukodwa ekuqiniseni, ekulondolozeni nasekwakheni amathambo.

 

Indima ye-S-4(Andarine)

I-S-4 inceda i-oxidize amafutha kwaye igcina umzimba kwi-catabolic ngexesha lokutya okuphantsi kweekhalori, eyona indima yayo ephambili.I-S-4 yenza izihlunu zibe nzima, zome, zichazwe ngakumbi kwaye zikhulise ukusabalalisa kwe-vascular.Inika inzuzo ebalulekileyo kumandla kunye nokunyamezela nakwiimeko zekhalori.Kwiidosi eziphezulu, kunokukhokelela ekuzuzeni ubunzima bomzimba obuthile.I-S-4 isoloko isetyenziselwa ukudibanisa nezinye i-SARMS kuba impembelelo yayo ekuzuzeni ubunzima bomzimba obunzima ayibalulekanga ngokwayo, nangona i-S-4 ingasetyenziselwa yodwa ngexesha lokulahlekelwa kwamafutha kwaye inike iziphumo ezigqwesileyo.

I-Estrogen: I-S-4 ayinayo i-aromatize kwi-estrogen kwaye ayinayo umsebenzi we-estrogenic wayo, ngaphandle kwemiphumo echaphazelekayo ehambelana ne-estrogen.

I-Androgen: I-S-4 ayinayo ipropathi ye-androgen kwaye ngoko ayinayo imiphumo emibi ye-androgen

I-Cardiovascular: I-S-4 ayinayo imiphumo emibi kwimpilo ye-cardiovascular health

I-Testosterone inhibition: I-S-4 ibonisa ukuvinjelwa okuncinci kakhulu kwiidosi eziphezulu, nangona kungekhona kakhulu njenge-LGD-4033, kodwa inhibition engaphezulu kune-MK-2886

I-Hepatotoxicity: I-S-4 ayinayo ityhefu esibindini.

 

Ukusetyenziswa kwe-S-4(Andarine)

I-dose yemihla ngemihla ephakanyisiweyo ye-S-4 yi-50-75mg, ukuya kwi-100mg ukuba umzimba wakho unokunyamezela, kodwa ndincoma ukuqala nge-dose ephantsi kunye nokwandisa ngokuthe ngcembe ukuphepha iziphumo ezingafunekiyo.I-S-4 inesiqingatha sobomi beeyure ze-4, ngoko thabatha ubuncinane kabini ngosuku, ngokukhethekileyo kwiidosi ezintathu, kwaye i-S4 isetyenziswe kakuhle ukuya kwiiveki ze-8, njengoko kungekho tyhefu yesibindi kwaye ixesha elide aliyingozi isibindi.


Ixesha lokuposa: Dec-23-2022