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Ipamorelin CAS: 170851-70-4 IPAMORELIN; AIB-HIS-D-NAL (2) -D-PHE-LYS-NH2

ibisobanuro bigufi:


  • URUBANZA OYA:170851-70-4
  • Izina:Ipamorelin
  • Uburemere bwa molekile:711.85
  • Imiti yimiti:C38H49N9O5
  • Ingingo yo gushonga:144-147 ° C.
  • Ingingo itetse:1185.5 ± 65.0 ° C (Biteganijwe)
  • ubucucike:1.263 ± 0.06 g / cm3 (Biteganijwe)
  • ububiko bwo kubika.:-20 ° C Ikonjesha
  • pka:13.04 ± 0.46 (Byahanuwe)
  • ifishi:ifu
  • Imisozi:711.868
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  • Ibicuruzwa birambuye

    Ibicuruzwa

    Ikoreshwa

    Ipamorelin (INN) (kode yiterambere NNC 26-0161) ni peptide-itoranya agonist ya auxin irekura peptide / reseptor ya somatosecretine (GHS) na somatosecretine.Ni pentapeptide hamwe na aside amine ikurikirana Aib-His-D-2-Nal - D-Phe -Lys-NH 2, ikomoka kuri GHRP-1.

    Ipamorelin yongerera cyane imisemburo ikura ya plasma (GH) mubikoko ndetse nabantu.Byongeye, ipamorelin yatumye ibiro byiyongera mubikoko.Kimwe na pralmorelin na GHRP-6, ipamorelin ntabwo igira ingaruka kuri prolactine, imisemburo itera imisemburo (FSH), imisemburo ya luteinizing (LH), cyangwa thyrotropine (TSH).Ariko, bitandukanye na pramoline (GHRP-2) na GHRP-6, ariko bisa na hormone yo gukura irekura imisemburo (GHRH), iparerelin ntabwo itera gusohora imisemburo ya adrenocorticotropique (ACTH) cyangwa cortisol kandi ihitamo cyane gutera ururenda rwa GH gusa.

    Ipamorelin yabanje gutunganywa na Novo Nordisk kandi ikora ibizamini byo mu cyiciro cya kabiri ubwacyo nk'umuti wa ilobstruction nyuma yo kubagwa, ariko byahagaritswe kubera kubura imikorere.

    Ipamorelin yakoreshejwe nabakinnyi nkibikorwa byongera ibiyobyabwenge.

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